The concept of structural medicinal chemistry would be applied during the course to study the drugs affecting cardiovascular system, antihistamines, histamine-release inhibitors, anti-ulcers, oral hypoglycaemic agents, centrally and peripherally acting analgesics, local anaesthetics, steroids and therapeutically related compounds classes. The concept will be applied through the comprehensive study of the relationship between drugs chemical structures (functional groups composition and 3D shape) and their pharmacodynamics and pharmacokinetic profiles.